SCHEMBL20005896

SCHEMBL20005896

CC(N)(CCO)c1ccccc1F

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 5/20 0.39
KCNE1 P15382 1/20 0.35
KCNQ1 P51787 1/20 0.35
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
KIF11 P52732 2/20 0.33
ALDH1A1 P00352 2/20 0.32
TSHR P16473 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CTNNB1 P35222 1/20 0.32
WNT3A P56704 1/20 0.32
ESR2 Q92731 1/20 0.32
TAAR1 Q96RJ0 2/20 0.31
SLC6A2 P23975 1/20 0.31
ACHE P22303 1/20 0.31
RIPK1 Q13546 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12077605 1.00 KCNN4 (0.39) KCNN4KCNE1KCNQ1HDAC3HDAC1
SCHEMBL17118587 0.89 KCNN4 (0.37) KCNN4KCNE1KCNQ1HDAC3HDAC1
SCHEMBL15536032 0.86 KCNN4 (0.42) KCNN4KCNE1KCNQ1HDAC3HDAC1
SCHEMBL15602054 0.86 KCNN4 (0.42) KCNN4KCNE1KCNQ1HDAC3HDAC1
Hydrochloric Acid SCHEMBL16833856 0.85 KCNN4 (0.41) KCNN4KCNE1KCNQ1HDAC3HDAC1
Hydrochloric Acid SCHEMBL18185126 0.85 KCNN4 (0.41) KCNN4KCNE1KCNQ1HDAC3HDAC1
SCHEMBL12077509 0.81 KCNN4 (0.35) KCNN4KCNE1KCNQ1HDAC3HDAC1
SCHEMBL434166 0.79 GABRA1 (0.38) ALDH1A1TSHRTDP1CTNNB1WNT3A
SCHEMBL21058252 0.79 KCNN4 (0.38) KCNN4KCNE1KCNQ1HDAC3HDAC1
SCHEMBL18683297 0.78 KCNN4 (0.39) KCNN4KCNE1KCNQ1KIF11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2864324-B1 DIFLUORO-HEXAHYDRO-CYCLOPENTAOXAZINYLS AND DIFLUORO-HEXAHYDRO-BENZOOXAZINYLS AS BACE1 INHIBITORS HOFFMANN LA ROCHE (CH) 2018-03-28 EP disclosed