SCHEMBL20006918

SCHEMBL20006918

CNc1ccc(-c2csc3c(-c4cnn(C)c4)cnc(N)c23)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 16/20 0.72
AURKB Q96GD4 12/20 0.72
AURKA O14965 7/20 0.72
MAP4K4 O95819 7/20 0.72
ABL1 P00519 7/20 0.72
NTRK1 P04629 7/20 0.72
INSR P06213 7/20 0.72
FYN P06241 7/20 0.72
LYN P07948 7/20 0.72
MET P08581 7/20 0.72
FGFR1 P11362 7/20 0.72
SRC P12931 7/20 0.72
BLK P51451 7/20 0.72
STK3 Q13188 7/20 0.72
NTRK2 Q16620 7/20 0.72
TAOK1 Q7L7X3 7/20 0.72
PLK4 O00444 6/20 0.72
CSF1R P07333 6/20 0.72
FLT1 P17948 6/20 0.72
RPS6KB1 P23443 6/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19996024 0.79 KDR (1.00) KDRAURKBAURKAMAP4K4ABL1
SCHEMBL14643163 0.78 KDR (0.60) KDRAURKBAURKAMAP4K4ABL1
SCHEMBL18590958 0.76 KDR (0.58) KDRAURKBAURKAMAP4K4ABL1
SCHEMBL10198705 0.75 KDR (0.57) KDRAURKBAURKAMAP4K4ABL1
SCHEMBL17034035 0.75 KDR (0.57) KDRAURKBAURKAMAP4K4ABL1
SCHEMBL3528912 0.73 BTK (0.61) KDRAURKBAURKAMAP4K4ABL1
SCHEMBL3378132 0.73 BTK (0.67) KDRAURKBAURKAMAP4K4ABL1
SCHEMBL5474567 0.72 KDR (0.66) KDRAURKBAURKAMAP4K4ABL1
SCHEMBL4821973 0.72 KDR (0.80) KDRAURKBAURKAMAP4K4ABL1
SCHEMBL4827643 0.72 KDR (0.80) KDRAURKBAURKAMAP4K4ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018058098-A1 COMPOUNDS AND METHODS FOR TREATING OR PREVENTING ALZHEIMER'S DISEASE YALE UNIVERSITY (US) 2018-03-29 WO disclosed