SCHEMBL20008446

SCHEMBL20008446

CCCCCCCC(CCCCC)c1ccno1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.39
CYP19A1 P11511 3/20 0.39
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 3/20 0.39
CYP2D6 P10635 1/20 0.39
NR1I2 O75469 1/20 0.37
SLC2A1 P11166 1/20 0.35
CSNK1E P49674 1/20 0.35
OPRM1 P35372 1/20 0.34
FAAH O00519 1/20 0.34
MGLL Q99685 1/20 0.34
SPHK1 Q9NYA1 2/20 0.34
KCNA5 P22460 1/20 0.33
KCNH2 Q12809 1/20 0.33
BDKRB2 P30411 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18842935 1.00 CYP1A2 (0.39) CYP1A2CYP19A1CYP2C9CYP2C19CYP2D6
SCHEMBL20442226 1.00 CYP1A2 (0.39) CYP1A2CYP19A1CYP2C9CYP2C19CYP2D6
SCHEMBL21210844 1.00 CYP1A2 (0.39) CYP1A2CYP19A1CYP2C9CYP2C19CYP2D6
SCHEMBL20214851 1.00 CYP1A2 (0.39) CYP1A2CYP19A1CYP2C9CYP2C19CYP2D6
SCHEMBL19853485 0.98 CYP1A2 (0.38) CYP1A2CYP19A1CYP2C9CYP2C19CYP2D6
SCHEMBL21164225 0.84 CYP1A2 (0.38) CYP1A2CYP19A1CYP2C9CYP2C19CYP2D6
SCHEMBL18583188 0.76 CYP2C9 (0.34) CYP1A2CYP19A1CYP2C9CYP2C19CYP2D6
SCHEMBL20008796 0.76 CYP2C9 (0.40) CYP1A2CYP19A1CYP2C9CYP2C19CYP2D6
SCHEMBL25543688 0.74 LMNA (0.37) CYP1A2CYP19A1CYP2C9CYP2C19CYP2D6
SCHEMBL25954461 0.71 NR1I2 (0.36) CYP19A1CYP2C9CYP2C19NR1I2SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10244756-B2 Fungicidal N-cycloalkyl-N-{[ortho-(1-substituted-cycloalkyl)heteroaryl]methyl}(thio)carboxamides BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2019-04-02 US disclosed
US-20180146670-A1 FUNGICIDAL N-CYCLOALKYL-N-{[ORTHO-(1-SUBSTITUTED-CYCLOALKYL)HETEROARYL]METHYL}(THIO)CARBOXAMIDES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-05-31 US disclosed
US-20180086735-A1 N-CYCLOALKYL-N-(BIHETEROCYCLYETHYLENE)-(THIO)CARBOXAMIDE DERIVATIVES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180086735-A1 N-CYCLOALKYL-N-(BIHETEROCYCLYETHYLENE)-(THIO)CARBOXAMIDE DERIVATIVES CBR3, CYP51A1, CBR1 CYP1A2 67/4885CYP19A1 1435/4885CYP2C9 17/4885
US-20180146670-A1 FUNGICIDAL N-CYCLOALKYL-N-{[ORTHO-(1-SUBSTITUTED-CYCLOALKYL)HETEROARYL]METHYL}(THIO)CARBOXAMIDES CBR3, CBR1, CYP51A1 CYP1A2 9/4885CYP19A1 366/4885CYP2C9 32/4885
US-10244756-B2 Fungicidal N-cycloalkyl-N-{[ortho-(1-substituted-cycloalkyl)heteroaryl]methyl}(thio)carboxamides CBR3, CBR1, CYP51A1 CYP1A2 9/4885CYP19A1 366/4885CYP2C9 32/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.