SCHEMBL20008946

SCHEMBL20008946

CC(C)N1C[C@@H]2C[C@H]1CN2Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.47
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13440371 1.00 SIGMAR1 (0.47) SIGMAR1MAPT
SCHEMBL5493931 0.84 SIGMAR1 (0.42) SIGMAR1MAPT
SCHEMBL16982000 0.83 SIGMAR1 (0.48) SIGMAR1MAPT
SCHEMBL20328234 0.80 SIGMAR1 (0.51) SIGMAR1MAPT
SCHEMBL5496487 0.80 SIGMAR1 (0.46) SIGMAR1MAPT
SCHEMBL23869439 0.79 SIGMAR1 (0.40) SIGMAR1MAPT
SCHEMBL6995832 0.79 SIGMAR1 (0.50) SIGMAR1MAPT
SCHEMBL8698904 0.79 SIGMAR1 (0.50) SIGMAR1MAPT
SCHEMBL11776188 0.79 SIGMAR1 (0.50) SIGMAR1MAPT
SCHEMBL9963408 0.79 LMNA (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10308614-B2 Therapeutic compounds and uses thereof GENENTECH, INC. (US) 2019-06-04 US disclosed
US-20180086720-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH, INC. (US) 2018-03-29 US disclosed
US-20180086720-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH, INC. (US) 2018-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10308614-B2 Therapeutic compounds and uses thereof SMARCC1, SMARCC2, SMARCA4 SIGMAR1 1928/4885MAPT 2011/4885
US-20180086720-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF SMARCC1, SMARCC2, SMARCA4 SIGMAR1 1928/4885MAPT 2011/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.