SCHEMBL2000962

SCHEMBL2000962

CC(C(=O)O)c1ccc(OCCCNC2=C(c3ccccc3)S(O)(O)N(C(C)(C)C)C2=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 3/20 0.38
TDP1 Q9NUW8 1/20 0.38
CA12 O43570 3/20 0.38
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA4 P22748 3/20 0.38
CA9 Q16790 3/20 0.38
GPR88 Q9GZN0 6/20 0.37
PTGS2 P35354 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 2/20 0.36
HTT P42858 2/20 0.36
KMT2A Q03164 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PTGER4 P35408 1/20 0.35
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
GAA P10253 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2000963 0.91 NR1H2 (0.41) ALDH1A1KDM4ETDP1CA12CA1
SCHEMBL2005055 0.90 PTGS1 (0.40) ALDH1A1KDM4ETDP1CA12CA1
SCHEMBL2000480 0.87 TSHR (0.45) ALDH1A1KDM4EL3MBTL1MEN1HTT
SCHEMBL2001772 0.85 MAPT (0.47) ALDH1A1KDM4ETDP1L3MBTL1MEN1
SCHEMBL2005056 0.81 PTGS1 (0.40) ALDH1A1KDM4ECA12CA1CA2
SCHEMBL1998245 0.81 NR1H2 (0.43) ALDH1A1KDM4ETDP1CA12CA1
SCHEMBL2005919 0.81 TBXAS1 (0.35) KDM4EKMT2A
SCHEMBL2000298 0.81 KMT2A (0.43) ALDH1A1KDM4EHTTKMT2AGAA
SCHEMBL2004216 0.80 MEN1 (0.36) ALDH1A1KDM4EL3MBTL1MEN1HTT
SCHEMBL2003669 0.79 ALDH1A1 (0.41) ALDH1A1KDM4EMEN1KMT2AMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960380-B2 Non-anilinic derivatives of isothiazol-3(2H)-one 1,1-dioxides as liver X receptor modulators ASTRAZENECA AB (SE) 2011-06-14 US disclosed