SCHEMBL20014752

SCHEMBL20014752

Brc1cccc2c1CSc1ccccc1C2

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.37
RYR2 Q92736 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ALOX15 P16050 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
GAA P10253 1/20 0.31
HSD17B3 P37058 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20014606 0.80 HTR2A (0.38) RYR2HPGD
SCHEMBL20014743 0.79 HSD17B3 (0.40) RYR2MEN1KMT2AALOX15TDP1
SCHEMBL20014517 0.79 MEN1 (0.43) RYR2MEN1KMT2AALOX15TDP1
SCHEMBL19329812 0.79 TRPA1 (0.41) TRPA1TDP1ALDH1A1HPGDGAA
SCHEMBL20015243 0.79 DRD2 (0.34) RYR2MEN1KMT2AALOX15TDP1
SCHEMBL10906067 0.78
SCHEMBL20015049 0.77 RYR2 (0.30) RYR2
SCHEMBL20829466 0.76 PRCP (0.41) MEN1KMT2AALOX15TDP1ALDH1A1
SCHEMBL20123771 0.75 TEAD1 (0.33) RYR2MEN1KMT2AALOX15TDP1
SCHEMBL20123457 0.75 DRD2 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2620436-B1 SUBSTITUTED POLYCYCLIC CARBAMOYL PYRIDONE DERIVATIVE PRODRUG SHIONOGI & CO (JP) 2018-05-09 EP disclosed
EP-2444400-B1 SUBSTITUTED POLYCYCLIC CARBAMOYLPYRIDONE DERIVATIVE SHIONOGI & CO (JP) 2018-03-28 EP disclosed