SCHEMBL20015989

SCHEMBL20015989

O=Cc1cnn2ccc(N3CCCCC3)nc12

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SMPD3 Q9NY59 17/20 0.63
PARP1 P09874 1/20 0.41
PIM1 P11309 1/20 0.40
PIM2 Q9P1W9 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20015889 0.99 SMPD3 (0.62) SMPD3PIM1PIM2IRAK4
SCHEMBL860108 0.87 SMPD3 (0.50) SMPD3PARP1IRAK4
SCHEMBL12979110 0.78 SMPD3 (0.51) SMPD3PIM1PIM2IRAK4
SCHEMBL861194 0.78 SMPD3 (0.51) SMPD3PIM1PIM2IRAK4
SCHEMBL861193 0.78 SMPD3 (0.51) SMPD3PIM1PIM2IRAK4
SCHEMBL19560147 0.78 SMPD3 (0.58) SMPD3IRAK4
SCHEMBL31259868 0.78 SMPD3 (1.00) SMPD3PARP1
SCHEMBL20015997 0.78 SMPD3 (0.68) SMPD3
SCHEMBL21996850 0.77 SMPD3 (0.63) SMPD3IRAK4
SCHEMBL19631256 0.76 SMPD3 (0.59) SMPD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299372-A1 INTERMEDIATE COMPOUNDS FOR THE PREPARATION OFSUBSTITUTED PYRAZOLO[1,5-A]PYRIMIDINE COMPOUNDS AS TRK KINASE INHIBITORS Array Biopharma, Inc. (US) 2018-03-28 EP disclosed