SCHEMBL20016619

SCHEMBL20016619

CCc1ccc([C@@H](CN)C(=O)Nc2ccc3cnccc3c2)cc1

nearest known ligand 0.82

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 20/20 0.82
ROCK1 Q13464 3/20 0.82
MYLK4 Q86YV6 1/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Netarsudil-M1 SCHEMBL21412824 0.90 ROCK2 (1.00) ROCK2ROCK1MYLK4
Netarsudil-M1 SCHEMBL30607237 0.90 ROCK2 (1.00) ROCK2ROCK1MYLK4
Netarsudil-M1 SCHEMBL21430354 0.90 ROCK2 (1.00) ROCK2ROCK1MYLK4
Netarsudil-M1 SCHEMBL30607241 0.90 ROCK2 (1.00) ROCK2ROCK1MYLK4
Netarsudil-M1 SCHEMBL9883166 0.90 ROCK2 (1.00) ROCK2ROCK1MYLK4
Netarsudil-M1 SCHEMBL30692376 0.90 ROCK2 (1.00) ROCK2ROCK1MYLK4
Netarsudil-M1 SCHEMBL30607238 0.90 ROCK2 (1.00) ROCK2ROCK1MYLK4
Netarsudil-M1 SCHEMBL111706 0.89 ROCK2 (0.98) ROCK2ROCK1MYLK4
SCHEMBL21412790 0.89 ROCK2 (1.00) ROCK2ROCK1MYLK4
SCHEMBL21430778 0.89 ROCK2 (1.00) ROCK2ROCK1MYLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9931336-B2 Combination therapy AERIE PHARMACEUTICALS, INC. (US) 2018-04-03 US disclosed