Netarsudil-M1

Netarsudil-M1

SCHEMBL30607237

NC[C@H](C(=O)Nc1ccc2cnccc2c1)c1ccc(CO)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 20/20 1.00
ROCK1 Q13464 3/20 1.00
MYLK4 Q86YV6 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Netarsudil-M1 SCHEMBL30692376 1.00 ROCK2 (1.00) ROCK2ROCK1MYLK4
Netarsudil-M1 SCHEMBL21412824 1.00 ROCK2 (1.00) ROCK2ROCK1MYLK4
Netarsudil-M1 SCHEMBL21430354 1.00 ROCK2 (1.00) ROCK2ROCK1MYLK4
Netarsudil-M1 SCHEMBL30607241 1.00 ROCK2 (1.00) ROCK2ROCK1MYLK4
Netarsudil-M1 SCHEMBL9883166 1.00 ROCK2 (1.00) ROCK2ROCK1MYLK4
Netarsudil-M1 SCHEMBL30607238 1.00 ROCK2 (1.00) ROCK2ROCK1MYLK4
Netarsudil-M1 SCHEMBL111706 0.99 ROCK2 (0.98) ROCK2ROCK1MYLK4
SCHEMBL20016619 0.90 ROCK2 (0.82) ROCK2ROCK1MYLK4
SCHEMBL23927626 0.89 ROCK2 (0.80) ROCK2ROCK1MYLK4
SCHEMBL13074858 0.89 ROCK2 (1.00) ROCK2ROCK1MYLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117050013-A Mono (acid) salts of 6-aminoisoquinolines and use thereof 爱瑞制药公司 2023-11-14 CN disclosed
CN-111936139-B Mono (acid) salts of 6-aminoisoquinolines and use thereof 爱瑞制药公司 2023-10-13 CN disclosed