SCHEMBL20018664

SCHEMBL20018664

NCc1cc(/C=C/C(=O)O)ccc1-c1ccc(O)c(C23CC4CC(CC(C4)C2)C3)c1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 9/20 0.73
NR0B2 Q15466 3/20 0.73
RARB P10826 6/20 0.70
HDAC11 Q96DB2 4/20 0.56
HDAC4 P56524 2/20 0.56
HDAC7 Q8WUI4 2/20 0.56
HDAC8 Q9BY41 2/20 0.56
HDAC6 Q9UBN7 2/20 0.56
HDAC9 Q9UKV0 2/20 0.56
HDAC3 O15379 1/20 0.56
HDAC2 Q92769 1/20 0.56
HDAC5 Q9UQL6 1/20 0.56
RARA P10276 3/20 0.52
RARG P13631 3/20 0.52
HDAC1 Q13547 1/20 0.47
HDAC10 Q969S8 1/20 0.47
PTPRCAP Q14761 1/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29462722 0.94 PTPN11 (0.66) PTPN11NR0B2RARBHDAC11HDAC4
SCHEMBL20018663 0.87 PTPN11 (0.56) PTPN11NR0B2RARBHDAC11HDAC4
SCHEMBL20018689 0.87 HDAC11 (0.59) PTPN11NR0B2RARBHDAC11HDAC4
SCHEMBL2389152 0.86 RARB (0.80) PTPN11NR0B2RARBHDAC11HDAC4
SCHEMBL2389155 0.86 RARB (0.80) PTPN11NR0B2RARBHDAC11HDAC4
SCHEMBL2393228 0.85 PTPN11 (0.71) PTPN11NR0B2RARBHDAC11HDAC4
SCHEMBL1914215 0.85 PTPN11 (1.00) PTPN11NR0B2RARBHDAC11HDAC4
SCHEMBL2391204 0.85 PTPN11 (0.77) PTPN11NR0B2RARBHDAC11HDAC4
SCHEMBL2407028 0.85 PTPN11 (0.77) PTPN11NR0B2RARBHDAC11HDAC4
SCHEMBL2391213 0.85 PTPN11 (0.77) PTPN11NR0B2RARBHDAC11HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3301085-A1 RETINOID DERIVATIVES WITH ANTITUMOR ACTIVITY BIOGEM S.CA.R.L. (IT) 2018-04-04 EP disclosed