SCHEMBL20018663

SCHEMBL20018663

CC1CC2CC(C1)CC(C)(c1cc(-c3ccc(/C=C/C(=O)O)cc3CN)ccc1O)C2

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 10/20 0.56
NR0B2 Q15466 4/20 0.56
RARB P10826 4/20 0.52
HDAC11 Q96DB2 3/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
RXRA P19793 1/20 0.41
AKR1B10 O60218 1/20 0.39
AKR1B1 P15121 1/20 0.39
AKR1C3 P42330 1/20 0.39
RARA P10276 1/20 0.38
RARG P13631 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20018664 0.87 PTPN11 (0.73) PTPN11NR0B2RARBHDAC11HDAC3
SCHEMBL20122014 0.85 RARB (0.72) PTPN11NR0B2RARBHDAC11HDAC3
Trifluoroacetic Acid SCHEMBL29462722 0.82 PTPN11 (0.66) PTPN11NR0B2RARBHDAC11HDAC3
SCHEMBL20018689 0.78 HDAC11 (0.59) PTPN11NR0B2RARBHDAC11HDAC4
SCHEMBL20122000 0.76 RARB (0.56) PTPN11NR0B2RARBHDAC11HDAC3
SCHEMBL2393228 0.74 PTPN11 (0.71) PTPN11NR0B2RARBHDAC11HDAC3
SCHEMBL2391204 0.74 PTPN11 (0.77) PTPN11NR0B2RARBHDAC11HDAC3
SCHEMBL2391213 0.74 PTPN11 (0.77) PTPN11NR0B2RARBHDAC11HDAC3
SCHEMBL20018658 0.74 PTPN11 (0.64) PTPN11NR0B2RARBHDAC11HDAC3
SCHEMBL2389152 0.73 RARB (0.80) PTPN11NR0B2RARBHDAC11HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3301085-A1 RETINOID DERIVATIVES WITH ANTITUMOR ACTIVITY BIOGEM S.CA.R.L. (IT) 2018-04-04 EP disclosed