SCHEMBL20020741

SCHEMBL20020741

Cc1cc2nc(C(=O)N(C)C)ccc2c(-c2ccc(Cl)cc2)c1[C@H](OC(C)(C)C)C(O)O

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.35
PSIP1 O75475 1/20 0.35
MALT1 Q9UDY8 1/20 0.34
CYP3A4 P08684 1/20 0.34
NPC1 O15118 1/20 0.33
DHODH Q02127 2/20 0.31
CNR1 P21554 1/20 0.31
PIK3CD O00329 1/20 0.30
PIK3CA P42336 1/20 0.30
PIK3CB P42338 1/20 0.30
PI4KA P42356 1/20 0.30
PIK3CG P48736 1/20 0.30
PI4KB Q9UBF8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL244670 0.87 PSIP1 (0.47) GRM2PSIP1MALT1CYP3A4DHODH
SCHEMBL243265 0.87 PSIP1 (0.47) GRM2PSIP1MALT1CYP3A4DHODH
SCHEMBL15182609 0.85 CYP3A4 (0.40) GRM2PSIP1MALT1CYP3A4NPC1
SCHEMBL3322579 0.85 PSIP1 (0.37) GRM2PSIP1MALT1CYP3A4NPC1
SCHEMBL20021129 0.82 MCHR1 (0.32) PSIP1CYP3A4
SCHEMBL247279 0.78 PSIP1 (0.43) GRM2PSIP1CYP3A4NPC1DHODH
SCHEMBL246062 0.78 PSIP1 (0.43) GRM2PSIP1CYP3A4NPC1DHODH
SCHEMBL20020744 0.78 TLR7 (0.33) PSIP1CYP3A4DHODH
SCHEMBL243122 0.77 PSIP1 (0.49) GRM2PSIP1CYP3A4DHODH
SCHEMBL243123 0.77 PSIP1 (0.49) GRM2PSIP1CYP3A4DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588455-B1 2-QUINOLINYL-ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES INC (US) 2018-04-04 EP disclosed