SCHEMBL20021185

SCHEMBL20021185

Cc1cc2nc(-c3cn[nH]c3)ccc2c(-c2ccc(Cl)cc2)c1C(OC(C)(C)C)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 1/20 0.45
CYP3A4 P08684 1/20 0.43
ROCK2 O75116 9/20 0.37
PRKD3 O94806 1/20 0.37
PRKCG P05129 1/20 0.37
PRKCB P05771 1/20 0.37
BRAF P15056 1/20 0.37
PRKCA P17252 1/20 0.37
PRKCH P24723 1/20 0.37
AKT1 P31749 1/20 0.37
PRKCI P41743 1/20 0.37
PRKCE Q02156 1/20 0.37
PRKCQ Q04759 1/20 0.37
PRKCZ Q05513 1/20 0.37
PRKCD Q05655 1/20 0.37
PRKD1 Q15139 1/20 0.37
ACACB O00763 1/20 0.35
ACACA Q13085 1/20 0.35
AKT2 P31751 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL251691 1.00 PSIP1 (0.45) PSIP1CYP3A4ROCK2PRKD3PRKCG
SCHEMBL15182665 0.93 PSIP1 (0.37) PSIP1CYP3A4ROCK2PRKD3PRKCG
SCHEMBL243700 0.91 PSIP1 (0.50) PSIP1CYP3A4
SCHEMBL10272175 0.89 CYP3A4 (0.46) PSIP1CYP3A4ROCK2PRKD3PRKCG
SCHEMBL3304151 0.88 PSIP1 (0.48) PSIP1CYP3A4
SCHEMBL244852 0.88 PSIP1 (0.46) PSIP1CYP3A4
SCHEMBL20021109 0.88 PSIP1 (0.46) PSIP1CYP3A4
SCHEMBL246425 0.86 PSIP1 (0.47) PSIP1CYP3A4
SCHEMBL20021158 0.86 PSIP1 (0.47) PSIP1CYP3A4
SCHEMBL245429 0.86 PSIP1 (0.45) PSIP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588455-B1 2-QUINOLINYL-ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES INC (US) 2018-04-04 EP disclosed