SCHEMBL3304151

SCHEMBL3304151

Cc1cc2nc(-c3ccccc3)ccc2c(-c2ccc(Cl)cc2)c1[C@H](OC(C)(C)C)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 1/20 0.48
CYP3A4 P08684 1/20 0.47
DHODH Q02127 3/20 0.40
MAPT P10636 3/20 0.39
TP53 P04637 1/20 0.39
THRB P10828 1/20 0.39
CTRC Q99895 1/20 0.39
TACR3 P29371 1/20 0.39
KDM4E B2RXH2 1/20 0.38
FABP3 P05413 1/20 0.38
FABP4 P15090 1/20 0.38
LTB4R Q15722 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL243700 0.97 PSIP1 (0.50) PSIP1CYP3A4DHODHMAPTTP53
SCHEMBL246425 0.93 PSIP1 (0.47) PSIP1CYP3A4DHODHMAPTKDM4E
SCHEMBL20021158 0.93 PSIP1 (0.47) PSIP1CYP3A4DHODHMAPTKDM4E
SCHEMBL245429 0.92 PSIP1 (0.45) PSIP1CYP3A4DHODHMAPTKDM4E
SCHEMBL247215 0.90 PSIP1 (0.45) PSIP1CYP3A4DHODHMAPTTACR3
SCHEMBL20021109 0.90 PSIP1 (0.46) PSIP1CYP3A4DHODHMAPTKDM4E
SCHEMBL244852 0.90 PSIP1 (0.46) PSIP1CYP3A4DHODHMAPTKDM4E
SCHEMBL15182560 0.89 PSIP1 (0.41) PSIP1CYP3A4DHODHMAPTTP53
SCHEMBL251691 0.88 PSIP1 (0.45) PSIP1CYP3A4
SCHEMBL20021185 0.88 PSIP1 (0.45) PSIP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012003498-A1 2 -QUINOLINYL- ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2012-01-05 WO disclosed