SCHEMBL20025375

SCHEMBL20025375

CCc1ccnc(N2CCOC3(CCN(Cc4cccc(CCOCCC(=O)OC(C)(C)C)c4Cl)CC3)C2)c1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 14/20 0.36
CHRM3 P20309 14/20 0.36
MGLL Q99685 1/20 0.33
EIF2AK4 Q9P2K8 1/20 0.32
P4HB P07237 1/20 0.32
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
FFAR1 O14842 1/20 0.31
METTL3 Q86U44 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20025020 0.92 MGLL (0.34) CHRM2CHRM3MGLLEIF2AK4PIK3CA
SCHEMBL20024916 0.89 CHRM2 (0.36) CHRM2CHRM3MGLLEIF2AK4P4HB
SCHEMBL20025496 0.84 CHRM2 (0.35) CHRM2CHRM3MGLLPIK3CDPIK3CA
SCHEMBL20025373 0.81 CHRM2 (0.32) CHRM2CHRM3FFAR1
SCHEMBL20025377 0.81 CHRM2 (0.38) CHRM2CHRM3MGLLP4HBFFAR1
SCHEMBL20025011 0.80 CHRM2 (0.39) CHRM2CHRM3MGLLP4HBFFAR1
SCHEMBL28688585 0.79 CHRM2 (0.38) CHRM2CHRM3MGLLFFAR1METTL3
SCHEMBL1246088 0.79 CHRM2 (0.60) CHRM2CHRM3
SCHEMBL12913087 0.77 CHRM2 (0.39) CHRM2CHRM3
SCHEMBL20025382 0.77 CHRM2 (0.37) CHRM2CHRM3MGLLFFAR1METTL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018059537-A1 DIAZASPIRO[5.5]UNDECANE DERIVATIVE AND USE THEREOF 四川海思科制药有限公司 2018-04-05 WO disclosed