SCHEMBL20024916

SCHEMBL20024916

CCc1ccnc(N2CCOC3(CCN(Cc4cccc(CCOCCC(=O)OC(C)(C)C)c4)CC3)C2)c1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 10/20 0.36
CHRM3 P20309 10/20 0.36
TBK1 Q9UHD2 1/20 0.34
METTL3 Q86U44 1/20 0.33
P4HB P07237 1/20 0.33
MGLL Q99685 2/20 0.32
FFAR1 O14842 2/20 0.32
EIF2AK4 Q9P2K8 1/20 0.32
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20025377 0.92 CHRM2 (0.38) CHRM2CHRM3TBK1METTL3P4HB
SCHEMBL20025011 0.91 CHRM2 (0.39) CHRM2CHRM3METTL3P4HBMGLL
SCHEMBL28688585 0.90 CHRM2 (0.38) CHRM2CHRM3METTL3MGLLFFAR1
SCHEMBL20025375 0.89 CHRM2 (0.36) CHRM2CHRM3METTL3P4HBMGLL
SCHEMBL20025020 0.89 MGLL (0.34) CHRM2CHRM3TBK1METTL3MGLL
SCHEMBL20025382 0.87 CHRM2 (0.37) CHRM2CHRM3METTL3MGLLFFAR1
SCHEMBL20025304 0.85 SIGMAR1 (0.41) DRD2DRD3
SCHEMBL20025288 0.84 SIGMAR1 (0.37) CHRM2CHRM3METTL3FFAR1DRD3
SCHEMBL20025335 0.84 CHRM2 (0.35) CHRM2CHRM3METTL3MGLLFFAR1
SCHEMBL20025290 0.83 SIGMAR1 (0.32) CHRM2CHRM3METTL3MGLLEIF2AK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018059537-A1 DIAZASPIRO[5.5]UNDECANE DERIVATIVE AND USE THEREOF 四川海思科制药有限公司 2018-04-05 WO disclosed