Phenylpiperazine

Phenylpiperazine

SCHEMBL2002893

NC(N)=O.c1ccc(N2CCNCC2)cc1

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 5/20 0.77
SIGMAR1 Q99720 4/20 0.77
HTR3E A5X5Y0 3/20 0.77
HTR3B O95264 3/20 0.77
HTR3A P46098 3/20 0.77
HTR3D Q70Z44 3/20 0.77
HTR3C Q8WXA8 3/20 0.77
USP2 O75604 3/20 0.67
ALDH1A1 P00352 3/20 0.67
TSHR P16473 2/20 0.67
HSD17B10 Q99714 1/20 0.67
HTR6 P50406 4/20 0.57
HTR1A P08908 2/20 0.56
HTR7 P34969 2/20 0.56
LTA4H P09960 1/20 0.56
CYP2D6 P10635 2/20 0.53
HTR2C P28335 2/20 0.53
TP53 P04637 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenylpiperazine SCHEMBL27922559 0.93 ADRB1 (0.71) ADRB1SIGMAR1HTR3EHTR3BHTR3A
Phenylpiperazine SCHEMBL11621472 0.92 ADRB1 (0.83) ADRB1SIGMAR1HTR3EHTR3BHTR3A
Phenylpiperazine SCHEMBL6495303 0.90 SIGMAR1 (0.67) ADRB1SIGMAR1HTR3EHTR3BHTR3A
Phenylpiperazine SCHEMBL29235064 0.90 TSHR (0.69) ADRB1SIGMAR1HTR3EHTR3BHTR3A
Phenylpiperazine SCHEMBL27606301 0.88 ADRB1 (0.91) ADRB1SIGMAR1HTR3EHTR3BHTR3A
Phenylpiperazine SCHEMBL29135595 0.88 ADRB1 (1.00) ADRB1SIGMAR1HTR3EHTR3BHTR3A
Phenylpiperazine SCHEMBL27858598 0.88 ADRB1 (1.00) ADRB1SIGMAR1HTR3EHTR3BHTR3A
Phenylpiperazine SCHEMBL55125 0.88 ADRB1 (1.00) ADRB1SIGMAR1HTR3EHTR3BHTR3A
Phenylpiperazine SCHEMBL24889 0.88 ADRB1 (1.00) ADRB1SIGMAR1HTR3EHTR3BHTR3A
Phenylpiperazine SCHEMBL4828251 0.86 ADRB1 (0.87) ADRB1SIGMAR1HTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7964605-B2 Phenyl piperazine compounds, pharmaceutical composition comprising the same, and use thereof SK HOLDINGS CO., LTD. (KR) 2011-06-21 US claimed
US-20090298851-A1 PHENYL PIPERAZINE COMPOUNDS, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME AND USE THEREOF SK BIOPHARMACEUTICALS CO., LTD. (KR) 2009-12-03 US claimed
WO-2009145590-A2 PHENYL PIPERAZINE COMPOUNDS, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME, AND USE THEREOF SK HOLDINGS CO., LTD. (KR) 2009-12-03 WO claimed
US-7964605-B2 Phenyl piperazine compounds, pharmaceutical composition comprising the same, and use thereof SK HOLDINGS CO., LTD. (KR) 2011-06-21 US disclosed
US-20090298851-A1 PHENYL PIPERAZINE COMPOUNDS, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME AND USE THEREOF SK BIOPHARMACEUTICALS CO., LTD. (KR) 2009-12-03 US disclosed
WO-2009145590-A2 PHENYL PIPERAZINE COMPOUNDS, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME, AND USE THEREOF SK HOLDINGS CO., LTD. (KR) 2009-12-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090298851-A1 PHENYL PIPERAZINE COMPOUNDS, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME AND USE THEREOF GRIK5, PLP2, PMP22 ADRB1 1434/4885SIGMAR1 526/4885HTR3E 1038/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.