SCHEMBL2003025

SCHEMBL2003025

COc1ccc2c(c1F)c(CC(=O)O)c(C)n2C(=O)N1CCCCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.42
AKR1C3 P42330 6/20 0.39
AKR1C2 P52895 6/20 0.39
LMNA P02545 3/20 0.37
CYP1A2 P05177 3/20 0.37
CYP2C9 P11712 3/20 0.37
NPSR1 Q6W5P4 3/20 0.37
CYP2D6 P10635 2/20 0.37
TSHR P16473 2/20 0.37
HIF1A Q16665 2/20 0.37
NFKB1 P19838 1/20 0.37
PTGS1 P23219 2/20 0.37
PTGS2 P35354 2/20 0.37
AKR1C4 P17516 2/20 0.36
AKR1C1 Q04828 2/20 0.36
PTGIR P43119 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 2/20 0.36
ABCB1 P08183 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2005243 0.91 AKR1C3 (0.39) CNR2AKR1C3AKR1C2LMNACYP1A2
SCHEMBL2007824 0.90 AKR1C3 (0.38) CNR2AKR1C3AKR1C2LMNACYP1A2
SCHEMBL2012093 0.87 CNR2 (0.42) CNR2AKR1C3AKR1C2LMNACYP1A2
SCHEMBL2006737 0.86 CNR2 (0.38) CNR2AKR1C3AKR1C2LMNACYP1A2
SCHEMBL2005335 0.82 AKR1C3 (0.39) AKR1C3AKR1C2LMNACYP1A2CYP2C9
SCHEMBL2004091 0.81 PTGS1 (0.48) CNR2AKR1C3AKR1C2LMNACYP1A2
SCHEMBL2009837 0.81 AKR1C3 (0.39) AKR1C3AKR1C2LMNACYP1A2CYP2C9
SCHEMBL2004524 0.81 AKR1C3 (0.39) AKR1C3AKR1C2LMNACYP1A2CYP2C9
SCHEMBL5549756 0.79 LMNA (0.59) AKR1C3AKR1C2LMNACYP1A2CYP2C9
SCHEMBL2002989 0.78 PTGDR2 (0.39) AKR1C3AKR1C2LMNACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed