SCHEMBL20030474

SCHEMBL20030474

CCc1c(C)cc2nc(-c3cnc4c(c3)c(N3CCN(C)CC3)cn4C)sc2c1-c1ccc(Cl)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CASP1 P29466 2/20 0.34
CASP7 P55210 2/20 0.34
HIF1A Q16665 2/20 0.34
HSD17B10 Q99714 2/20 0.34
ALDH1A1 P00352 1/20 0.34
GLA P06280 1/20 0.34
TNK2 Q07912 1/20 0.33
HRH4 Q9H3N8 3/20 0.33
BRD4 O60885 2/20 0.32
MCHR1 Q99705 1/20 0.32
MET P08581 1/20 0.31
SLC6A9 P48067 1/20 0.31
KCNH2 Q12809 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
HTR3A P46098 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906158 0.90 KDM4E (0.34) USP2CYP1A2CYP3A4CASP1CASP7
SCHEMBL31114924 0.81 MEN1 (0.34) ALDH1A1HRH4BRD4MCHR1MEN1
SCHEMBL20101207 0.81 MEN1 (0.34) ALDH1A1HRH4BRD4MCHR1MEN1
SCHEMBL15342181 0.80
SCHEMBL22506323 0.80 PSIP1 (0.36) CYP3A4BRD4KCNH2
SCHEMBL15342590 0.80 PSIP1 (0.36) CYP3A4BRD4KCNH2
SCHEMBL19906155 0.79 EIF4EBP1 (0.34) HRH4MCHR1MEN1MAPK10KMT2A
SCHEMBL20030685 0.77 KDM4E (0.33) ALDH1A1MCHR1MEN1KMT2AKDM4E
SCHEMBL19905935 0.74 KDM4E (0.34) ALDH1A1BRD4MEN1KMT2AKDM4E
SCHEMBL20030734 0.74 KDM4E (0.36) CYP1A2HSD17B10ALDH1A1BRD4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018064080-A1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING HIV INFECTION GILEAD SCIENCES, INC. (US) 2018-04-05 WO disclosed