SCHEMBL20030864

SCHEMBL20030864

CCOC(=O)Cc1c(C)cc2nc(-c3cnc4c(n3)c(N)nn4C)sc2c1-c1ccc(Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.42
TDP1 Q9NUW8 3/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.39
ALDH1A1 P00352 6/20 0.39
HPGD P15428 4/20 0.39
HTT P42858 3/20 0.39
RAB9A P51151 4/20 0.38
LMNA P02545 3/20 0.38
NPC1 O15118 3/20 0.38
TSHR P16473 2/20 0.38
POLB P06746 1/20 0.38
MEN1 O00255 5/20 0.38
KMT2A Q03164 5/20 0.38
MAPT P10636 4/20 0.38
MAPK1 P28482 1/20 0.37
FPR1 P21462 1/20 0.37
HSD17B10 Q99714 2/20 0.35
TP53 P04637 1/20 0.35
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20030762 0.85 KDM4E (0.38) KDM4ETDP1L3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL31114886 0.83 ALDH1A1 (0.36) KDM4ETDP1SMN1; SMN2ALDH1A1HPGD
SCHEMBL20101221 0.83 ALDH1A1 (0.36) KDM4ETDP1SMN1; SMN2ALDH1A1HPGD
SCHEMBL20030971 0.82 KDM4E (0.35) KDM4ETDP1L3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL20030866 0.82 KDM4E (0.35) KDM4ETDP1L3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL20030764 0.81 KDM4E (0.34) KDM4ETDP1L3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL20030995 0.81 KDM4E (0.43) KDM4ETDP1L3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL20030863 0.78 HTT (0.31) KDM4EALDH1A1HPGDHTT
SCHEMBL20030973 0.76 KDM4E (0.43) KDM4ETDP1L3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL20031011 0.76 KDM4E (0.38) KDM4ETDP1L3MBTL1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018064080-A1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING HIV INFECTION GILEAD SCIENCES, INC. (US) 2018-04-05 WO disclosed