SCHEMBL20031654

SCHEMBL20031654

CCOOc1ccc2c(c1)CCc1c(C#N)c(C#N)c3c(c1-2)-c1ccc(O)cc1CC3

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.40
MIF P14174 5/20 0.36
MAPK1 P28482 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
ALOX12 P18054 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ESR1 P03372 4/20 0.35
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
AKR1B1 P15121 1/20 0.33
CYP26A1 O43174 1/20 0.32
ESR2 Q92731 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25016883 0.83 EGFR (0.42) EGFRMIFMAPK1LMNASMN1; SMN2
SCHEMBL20031659 0.83 MIF (0.44) EGFRMIFMAPK1KDM4EALDH1A1
SCHEMBL22683261 0.81 MEN1 (0.46) EGFRMIFALDH1A1
SCHEMBL20031910 0.80 EGFR (0.44) EGFRMAPK1KDM4EALDH1A1LMNA
SCHEMBL22683259 0.77 BRD4 (0.48) MIFKDM4EALDH1A1FNTAFNTB
SCHEMBL20031875 0.76 EGFR (0.51) EGFRMAPK1KDM4EALDH1A1SMN1; SMN2
SCHEMBL20031646 0.76 EGFR (0.58) EGFRMAPK1KDM4EALDH1A1
SCHEMBL22703046 0.76 EGFR (0.44) EGFRMIFMAPK1KDM4EALDH1A1
SCHEMBL22683257 0.75 MAOB (0.39) EGFRMIFALDH1A1
SCHEMBL20031639 0.75 ALB (0.44) AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018063105-A1 [5]HELICENE DERIVATIVES AS MOLECULAR REPORTERS FOR DIAGNOSTIC APPLICATIONS AND METHODS OF SYNTHESIS THEREFOR NATIONAL SCIENCE AND TECHNOLOGY DEVELOPMENT AGENCY (TH) 2018-04-05 WO disclosed