SCHEMBL20031875

SCHEMBL20031875

CCOc1ccc2c(c1)CCc1c(C#N)c(C#N)c3c(c1-2)-c1ccc(OC)cc1CC3

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.51
MAPK1 P28482 1/20 0.47
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
MPO P05164 1/20 0.43
KDM4E B2RXH2 4/20 0.42
ALDH1A1 P00352 3/20 0.42
GLA P06280 1/20 0.42
CYP19A1 P11511 2/20 0.39
CYP11B1 P15538 2/20 0.39
CYP11B2 P19099 2/20 0.39
MAPT P10636 3/20 0.39
HTT P42858 1/20 0.39
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
MEN1 O00255 1/20 0.38
ALPL P05186 1/20 0.38
CLK1 P49759 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20031910 0.95 EGFR (0.44) EGFRMAPK1KDM4EALDH1A1GLA
SCHEMBL20031646 0.91 EGFR (0.58) EGFRMAPK1CYP1A2CYP2D6MPO
SCHEMBL20031900 0.85 EGFR (0.53) EGFRMAPK1CYP1A2CYP2D6MPO
SCHEMBL22702989 0.81 THRA (0.47) EGFRKDM4EALDH1A1MAPTHTT
SCHEMBL20031909 0.78 MAOB (0.43) EGFRMAPK1
SCHEMBL25017016 0.78 BRD4 (0.57) EGFRMAPK1KDM4EALDH1A1MAPT
SCHEMBL22703046 0.77 EGFR (0.44) EGFRMAPK1CYP1A2CYP2D6KDM4E
SCHEMBL22683261 0.76 MEN1 (0.46) EGFRALDH1A1MAPTMEN1KMT2A
SCHEMBL22683256 0.76 BRD4 (0.53) EGFRKDM4EMAPT
SCHEMBL20031911 0.74 MAOB (0.41) EGFRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018063105-A1 [5]HELICENE DERIVATIVES AS MOLECULAR REPORTERS FOR DIAGNOSTIC APPLICATIONS AND METHODS OF SYNTHESIS THEREFOR NATIONAL SCIENCE AND TECHNOLOGY DEVELOPMENT AGENCY (TH) 2018-04-05 WO disclosed