SCHEMBL2003393

SCHEMBL2003393

COc1ccc2c(c1)c(C(=O)c1ncc(-c3cccnc3)o1)c(Cl)n2Cc1ccc(Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.43
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43
RGS12 O14924 1/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
PKM P14618 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
MAPK1 P28482 1/20 0.43
CYP2C19 P33261 1/20 0.43
GNAI1 P63096 1/20 0.43
PMP22 Q01453 1/20 0.43
KMT2A Q03164 1/20 0.43
HIF1A Q16665 1/20 0.43
TNIK Q9UKE5 1/20 0.42
ALOX5 P09917 1/20 0.42
ALOX5AP P20292 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2005691 0.93 ALOX5AP (0.43) CYP3A4ALDH1A1LMNAMAPTCYP2C9
SCHEMBL2009799 0.93 PLA2G2A (0.49) CYP3A4ALDH1A1MEN1RGS12LMNA
SCHEMBL2003596 0.92 PLA2G2A (0.48) CYP3A4ALDH1A1MEN1RGS12LMNA
SCHEMBL2005733 0.91 MEN1 (0.45) CYP3A4ALDH1A1MEN1RGS12LMNA
SCHEMBL2000331 0.91 PTGES2 (0.41) CYP3A4ALDH1A1MEN1LMNAMAPT
SCHEMBL2003366 0.91 TP53 (0.39) CYP3A4ALDH1A1MAPTTNIKPLA2G2A
SCHEMBL2004581 0.90 ALOX5AP (0.41) CYP3A4ALDH1A1MEN1RGS12LMNA
SCHEMBL2005285 0.89 PTGES2 (0.43) ALDH1A1MEN1MAPTKMT2AALOX5
SCHEMBL2004090 0.88 PTGES2 (0.40) CYP3A4ALDH1A1MEN1LMNAMAPT
SCHEMBL2001738 0.88 CYP3A4 (0.44) CYP3A4ALDH1A1MEN1RGS12LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed