SCHEMBL2000331

SCHEMBL2000331

O=C(c1ncc(-c2cccnc2)o1)c1c(Cl)n(Cc2ccc(Cl)cc2)c2ccc(Cl)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 1/20 0.41
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
ALOX15 P16050 2/20 0.39
ALOX12 P18054 2/20 0.39
HSD17B10 Q99714 2/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
FAAH O00519 1/20 0.38
HDAC6 Q9UBN7 3/20 0.38
HDAC1 Q13547 2/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
TBXAS1 P24557 1/20 0.38
ALOX5 P09917 1/20 0.37
ALOX5AP P20292 1/20 0.37
MEN1 O00255 1/20 0.37
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004090 0.94 PTGES2 (0.40) PTGES2KDM4EALDH1A1MAPTALOX15
SCHEMBL2005285 0.93 PTGES2 (0.43) PTGES2KDM4EALDH1A1MAPTALOX15
SCHEMBL2001251 0.92 HDAC6 (0.42) PTGES2KDM4EALDH1A1MAPTALOX15
SCHEMBL2003393 0.91 CYP3A4 (0.43) PTGES2KDM4EALDH1A1MAPTHPGD
SCHEMBL2005326 0.91 MEN1 (0.43) PTGES2KDM4EALDH1A1MAPTALOX15
SCHEMBL2009494 0.90 FAAH (0.37) PTGES2KDM4EALDH1A1MAPTALOX12
SCHEMBL2005691 0.90 ALOX5AP (0.43) PTGES2KDM4EALDH1A1MAPTALOX15
SCHEMBL2010345 0.90 MEN1 (0.38) PTGES2MAPTALOX15ALOX12HSD17B10
SCHEMBL2002134 0.89 PTGES2 (0.42) PTGES2KDM4EALDH1A1MAPTALOX15
SCHEMBL2001640 0.86 L3MBTL1 (0.39) PTGES2KDM4EALDH1A1MAPTALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed