SCHEMBL20034085

SCHEMBL20034085

CC(C)(C)NC(O)c1cccc(-c2cnc3[nH]c(-c4ccccc4)cc3c2)n1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.45
ULK1 O75385 9/20 0.43
PIK3CG P48736 1/20 0.39
KIT P10721 6/20 0.39
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
RIPK1 Q13546 1/20 0.36
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20034116 0.79 BRD4 (0.41) BRD4ULK1PIK3CGKITCCNB2
SCHEMBL23912153 0.77 BRD4 (0.57) BRD4ULK1PIK3CGKITCCNB2
SCHEMBL18918755 0.77 ULK1 (0.60) BRD4ULK1PIK3CGKITRIPK1
SCHEMBL20034104 0.75 BRD4 (0.41) BRD4ULK1PIK3CGKITCCNB2
SCHEMBL20034111 0.75 BRD4 (0.40) BRD4ULK1PIK3CGKITCCNB2
SCHEMBL18944010 0.74 BRD4 (0.51) BRD4ULK1PIK3CGKITCCNB2
SCHEMBL18918667 0.74 ULK1 (0.59) BRD4ULK1PIK3CGKIT
SCHEMBL20034086 0.73 BRD4 (0.40) BRD4ULK1PIK3CGKITCCNB2
SCHEMBL20034087 0.73 BRD4 (0.41) BRD4ULK1PIK3CGKITCCNB2
SCHEMBL20034134 0.73 BRD4 (0.41) BRD4ULK1PIK3CGKITCCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9938273-B2 Compounds and methods for kinase modulation, and indications therefor PLEXXIKON INC. (US) 2018-04-10 US disclosed