SCHEMBL20034087

SCHEMBL20034087

CN(C1CCNC1)C(O)c1cccc(-c2cnc3[nH]c(-c4ccccc4)cc3c2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.41
ULK1 O75385 2/20 0.36
KIT P10721 6/20 0.35
PIK3CG P48736 1/20 0.34
SLC6A2 P23975 5/20 0.33
SLC6A4 P31645 5/20 0.33
SLC6A3 Q01959 3/20 0.33
CYP2D6 P10635 2/20 0.33
KCNH2 Q12809 2/20 0.33
CCNB2 O95067 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
CDK5 Q00535 1/20 0.33
CDK5R1 Q15078 1/20 0.33
CCNB3 Q8WWL7 1/20 0.33
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
NRAS P01111 1/20 0.33
FLT3 P36888 1/20 0.33
CHEK2 O96017 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18918820 0.81 ULK1 (0.46) BRD4ULK1KITPIK3CGSLC6A2
SCHEMBL18918838 0.74 ULK1 (0.51) BRD4ULK1KITPIK3CGRIPK1
SCHEMBL20034104 0.73 BRD4 (0.41) BRD4ULK1KITPIK3CGCCNB2
SCHEMBL20034116 0.73 BRD4 (0.41) BRD4ULK1KITPIK3CGCCNB2
SCHEMBL20034085 0.73 BRD4 (0.45) BRD4ULK1KITPIK3CGCCNB2
SCHEMBL18918839 0.72 ULK1 (0.51) BRD4ULK1KITRIPK1
SCHEMBL20034086 0.72 BRD4 (0.40) BRD4ULK1KITPIK3CGCCNB2
SCHEMBL20034101 0.72 BRD4 (0.41) BRD4ULK1KITPIK3CGKCNH2
SCHEMBL20034134 0.72 BRD4 (0.41) BRD4ULK1KITPIK3CGKCNH2
SCHEMBL20034117 0.71 BRD4 (0.39) BRD4ULK1KITPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9938273-B2 Compounds and methods for kinase modulation, and indications therefor PLEXXIKON INC. (US) 2018-04-10 US disclosed