SCHEMBL20034539

SCHEMBL20034539

C/C=C(\C)CC(=O)Bc1nnc(CCCCc2nnc(NC(=O)C/C(C)=C/C)s2)s1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GLS O94925 18/20 0.48
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19920381 0.88 GLS (0.59) GLSALDH1A1TSHR
SCHEMBL19920384 0.82 GLS (0.53) GLSALDH1A1TSHR
SCHEMBL19920154 0.80 GLS (0.63) GLSALDH1A1TSHR
SCHEMBL15727706 0.70 GLS (0.73) GLSALDH1A1TSHR
SCHEMBL15727679 0.69 GLS (0.68) GLSALDH1A1
SCHEMBL15748909 0.69 GLS (0.59) GLS
SCHEMBL15727776 0.67 GLS (0.76) GLSALDH1A1TSHR
SCHEMBL15727709 0.67 NPC1 (0.69) GLSALDH1A1
SCHEMBL15727702 0.67 GLS (0.64) GLSALDH1A1
SCHEMBL19920338 0.67 GLS (0.68) GLSALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9938267-B2 Heterocyclic inhibitors of glutaminase CALITHERA BIOSCIENCES, INC. (US) 2018-04-10 US disclosed