SCHEMBL20037042

SCHEMBL20037042

Cc1[nH]c2ccccc2c1CC(=O)OCC(=O)Cl

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK6 Q92876 4/20 0.61
KDM4E B2RXH2 6/20 0.61
ALDH1A1 P00352 5/20 0.61
MAPT P10636 3/20 0.61
GAA P10253 1/20 0.61
CASP1 P29466 1/20 0.61
CASP7 P55210 1/20 0.61
PRSS1 P07477 2/20 0.55
PRSS2 P07478 2/20 0.55
PRSS3 P35030 2/20 0.55
KLK7 P49862 1/20 0.55
KLK14 Q9P0G3 1/20 0.55
KLK5 Q9Y337 1/20 0.55
LMNA P02545 2/20 0.53
TSHR P16473 1/20 0.49
HTT P42858 1/20 0.49
EGFR P00533 2/20 0.48
POLB P06746 1/20 0.48
SLC2A1 P11166 1/20 0.47
CYP3A4 P08684 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20037329 0.88 MAPT (0.71) KLK6KDM4EALDH1A1MAPTGAA
SCHEMBL31487317 0.86 KDM4E (0.68) KLK6KDM4EALDH1A1MAPTGAA
SCHEMBL1165573 0.86 KDM4E (0.68) KLK6KDM4EALDH1A1MAPTGAA
SCHEMBL7877546 0.84 MAPT (0.73) KLK6KDM4EALDH1A1MAPTGAA
SCHEMBL20037195 0.82 MAPT (0.59) KLK6KDM4EALDH1A1MAPTGAA
SCHEMBL1191332 0.81 KDM4E (0.69) KLK6KDM4EALDH1A1MAPTGAA
SCHEMBL20037242 0.81 KLK6 (0.65) KLK6KDM4EALDH1A1MAPTGAA
SCHEMBL20037245 0.81 KDM4E (0.61) KLK6KDM4EALDH1A1MAPTGAA
SCHEMBL5643293 0.81 ALDH1A1 (0.65) KLK6KDM4EALDH1A1MAPTGAA
SCHEMBL20037094 0.81 KDM4E (0.61) KLK6KDM4EALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018065607-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2018-04-12 WO disclosed
EP-3305781-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN-RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum (DE) 2018-04-11 EP disclosed