SCHEMBL20037151

SCHEMBL20037151

Cc1nn(-c2ccc(C(F)(F)F)cc2)c(C)c1N

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.62
BRAF P15056 2/20 0.46
ALDH1A1 P00352 1/20 0.41
XDH P47989 1/20 0.41
SRC P12931 1/20 0.41
KDR P35968 1/20 0.41
NPY5R Q15761 1/20 0.40
ATM Q13315 1/20 0.40
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NR3C1 P04150 4/20 0.39
P2RX7 Q99572 1/20 0.38
CYP2C9 P11712 1/20 0.38
PTGS2 P35354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22632995 0.81 SMN1; SMN2 (0.59) SMN1; SMN2ALDH1A1NPY5RMAPTRAB9A
SCHEMBL11652228 0.81 SMN1; SMN2 (0.68) SMN1; SMN2BRAFSRCKDRRAB9A
SCHEMBL20037041 0.80 SMN1; SMN2 (0.72) SMN1; SMN2ALDH1A1MAPTRAB9AL3MBTL1
Water SCHEMBL11654225 0.79 SMN1; SMN2 (0.70) SMN1; SMN2ALDH1A1MAPTRAB9AL3MBTL1
SCHEMBL6966371 0.77 SMN1; SMN2 (1.00) SMN1; SMN2ALDH1A1MAPTRAB9A
SCHEMBL14353348 0.77 CYP1A2 (0.62) SMN1; SMN2BRAFALDH1A1NPY5RMAPT
SCHEMBL5904547 0.76 P2RX7 (0.46) SMN1; SMN2BRAFALDH1A1RAB9ANR3C1
SCHEMBL5904541 0.76 P2RX7 (0.46) BRAFATMRAB9ANR3C1P2RX7
SCHEMBL5904596 0.76 BRAF (0.43) BRAFNPY5RATMNR3C1CYP2C9
Water SCHEMBL11653913 0.76 SMN1; SMN2 (0.66) SMN1; SMN2ALDH1A1ATMMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018065607-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2018-04-12 WO disclosed
EP-3305781-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN-RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum (DE) 2018-04-11 EP disclosed