SCHEMBL2003729

SCHEMBL2003729

COc1ccc2c(c1)c(C(=O)c1nc(-c3cccnc3)co1)cn2Cc1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.47
ALDH1A1 P00352 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
MAPT P10636 2/20 0.44
AHR P35869 1/20 0.42
SERPINE1 P05121 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
CYP17A1 P05093 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
KDM4E B2RXH2 1/20 0.41
NPY1R P25929 1/20 0.41
HTT P42858 1/20 0.41
NPY2R P49146 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PTGS2 P35354 2/20 0.40
PLA2G2A P14555 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2006741 0.92 LMNA (0.54) LMNAALDH1A1SMN1; SMN2MAPTAHR
SCHEMBL2006991 0.91 LMNA (0.47) LMNAALDH1A1SMN1; SMN2MAPTAHR
SCHEMBL2008723 0.87 LMNA (0.49) LMNAALDH1A1SMN1; SMN2MAPTAHR
SCHEMBL2004312 0.86 LMNA (0.46) LMNAALDH1A1SMN1; SMN2MAPTAHR
SCHEMBL2003054 0.86 LMNA (0.51) LMNAALDH1A1SMN1; SMN2MAPTAHR
SCHEMBL2007318 0.85 LMNA (0.47) LMNAALDH1A1SMN1; SMN2MAPTAHR
SCHEMBL4083410 0.85 PDE4A (0.47) LMNAALDH1A1SMN1; SMN2MAPTSERPINE1
SCHEMBL2002672 0.85 LMNA (0.48) LMNAALDH1A1SMN1; SMN2MAPTAHR
SCHEMBL2000164 0.84 AHR (0.50) LMNAALDH1A1SMN1; SMN2MAPTAHR
SCHEMBL2006000 0.84 LMNA (0.48) LMNAALDH1A1SMN1; SMN2MAPTAHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed