SCHEMBL20037588

SCHEMBL20037588

C=C(C)c1ccc(N2CCC(C(=O)O)CC2)cn1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 9/20 0.46
KDM4E B2RXH2 2/20 0.46
CYP2C19 P33261 1/20 0.46
USP2 O75604 1/20 0.43
HPGD P15428 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD17B10 Q99714 1/20 0.43
AKR1C3 P42330 1/20 0.42
SYK P43405 1/20 0.42
HRH3 Q9Y5N1 3/20 0.42
NEK2 P51955 2/20 0.42
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22629266 0.83 HRH3 (0.58) NOTUMKDM4ECYP2C19USP2HPGD
SCHEMBL237457 0.81 KDM4E (0.55) NOTUMKDM4ECYP2C19USP2HPGD
SCHEMBL20037680 0.77 NOTUM (0.50) NOTUMKDM4ECYP2C19USP2HPGD
SCHEMBL16398202 0.77 NEK2 (0.52) NOTUMKDM4ECYP2C19USP2HPGD
SCHEMBL20207616 0.77 HDAC3 (0.46) KDM4ECYP2C19
SCHEMBL23114831 0.77 PRMT5 (0.47) NOTUMKDM4ECYP2C19USP2HPGD
SCHEMBL1441410 0.77 CHRNB2 (0.54) NOTUMKDM4ECYP2C19USP2HPGD
SCHEMBL20249117 0.77 HRH3 (0.49) NOTUMKDM4ECYP2C19USP2HPGD
SCHEMBL25146908 0.77 ACACB (0.49) NOTUMKDM4ECYP2C19USP2HPGD
SCHEMBL23103150 0.77 NOTUM (0.49) NOTUMKDM4ECYP2C19USP2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305785-A1 PYRIDO[3,4-d]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Teijin Pharma Limited (JP) 2018-04-11 EP disclosed