SCHEMBL20037598

SCHEMBL20037598

CNc1ccc(CN2[C@@H](C)COC[C@@H]2C)cn1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.39
GRM2 Q14416 1/20 0.39
ALDH1A1 P00352 1/20 0.35
CNR2 P34972 3/20 0.33
CDK4 P11802 2/20 0.33
CCND3 P30281 2/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
HCAR3 P49019 1/20 0.33
CDK6 Q00534 1/20 0.33
CPB2 Q96IY4 1/20 0.33
METTL3 Q86U44 1/20 0.33
NNMT P40261 1/20 0.33
CHEK1 O14757 1/20 0.32
ACHE P22303 1/20 0.32
AKT1 P31749 1/20 0.31
PIK3CA P42336 1/20 0.31
XIAP P98170 2/20 0.31
BIRC2 Q13490 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20037820 0.81 GRM2 (0.38) GRM2ALDH1A1
SCHEMBL2233826 0.79 GRM2 (0.38) MTORGRM2ALDH1A1
SCHEMBL20255421 0.79 GRM2 (0.38) GRM2ALDH1A1
SCHEMBL18291601 0.79 DRD2 (0.41) MTORGRM2ALDH1A1PIK3CA
SCHEMBL2233831 0.79 DRD2 (0.41) MTORGRM2ALDH1A1PIK3CA
SCHEMBL20249172 0.77 CCR9 (0.37) GRM2ALDH1A1
SCHEMBL23768076 0.74 HCAR3 (0.38) ALDH1A1CYP11B1CYP11B2HCAR3CPB2
SCHEMBL17828163 0.72 HRH3 (0.55) ALDH1A1METTL3ACHE
SCHEMBL171824 0.72 KMT2A (0.43) ALDH1A1
SCHEMBL27896110 0.71 GRM2 (0.35) GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305785-A1 PYRIDO[3,4-d]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Teijin Pharma Limited (JP) 2018-04-11 EP disclosed