SCHEMBL20039909

SCHEMBL20039909

CCOC(=O)C(N)C(=O)c1ccc(Oc2ccccc2)cc1C(C)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
HPGD P15428 1/20 0.44
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
SCN9A Q15858 1/20 0.43
PTGS2 P35354 2/20 0.42
ALDH1A1 P00352 4/20 0.39
MAPT P10636 3/20 0.39
ACACB O00763 2/20 0.39
ACACA Q13085 2/20 0.39
LMNA P02545 2/20 0.39
SRD5A2 P31213 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
THRB P10828 1/20 0.39
POLB P06746 1/20 0.39
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21065440 0.86 PTGS1 (0.44) HPGDALDH1A1ACACBACACASMN1; SMN2
SCHEMBL16613203 0.80 NPC1 (0.51) NPC1RAB9AHPGDCRHBPCRHR2
Hydrochloric Acid SCHEMBL16597575 0.79 NPC1 (0.50) NPC1RAB9AHPGDCRHBPCRHR2
SCHEMBL22447136 0.75 POLB (0.64) RAB9AHPGDALDH1A1MAPTLMNA
SCHEMBL23052920 0.72 NR1H4 (0.56) NPC1RAB9AHPGDMAPTLMNA
SCHEMBL9458638 0.72 SRD5A2 (0.54) NPC1RAB9AHPGDMAPTSRD5A2
SCHEMBL22447135 0.72 XDH (0.51) HPGDALDH1A1ACACBACACASMN1; SMN2
SCHEMBL31059195 0.72 NPC1 (0.54) NPC1RAB9AHPGDCRHBPCRHR2
SCHEMBL20630947 0.71 ALDH1A1 (0.45) RAB9AHPGDALDH1A1MAPTACACB
SCHEMBL13431425 0.71 TSHR (0.50) NPC1RAB9AALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305769-A1 METHOD FOR PREPARATION OF (7-PHENOXY-4-HYDROXY-1-METHYL-ISOQUINOLINE-3-CARBONYL)-GLYCINE (ROXEDUSTAT) AND ITS INTERMEDIATES BASED ON SIMULTANEOUS OPENING OF OXAZOLIC RING, FISSION OF ETHER AND CREATION OF IMINE Zentiva K.S. (CZ) 2018-04-11 EP disclosed