SCHEMBL20042649

SCHEMBL20042649

CN(C)c1nc(C2CC2)nc2c1CNC2

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.36
HTR2C P28335 6/20 0.36
HTR2B P41595 6/20 0.36
PDE10A Q9Y233 7/20 0.35
CHRM3 P20309 3/20 0.30
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042774 0.75 TUBB3 (0.34) HTR2C
SCHEMBL20042648 0.71 CHRM3 (0.51) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL2806533 0.65 LRRK2 (0.38)
SCHEMBL21035571 0.64 HTR2C (0.47) HTR2AHTR2CHTR2BPDE10ACHRM3
SCHEMBL20042975 0.63 CHRM3 (0.42) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL18649181 0.62 LMNA (0.50) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL22344966 0.62 HTR2C (0.32) HTR2CHTR2B
SCHEMBL14483195 0.61 HTR2C (0.32) HTR2AHTR2CHTR2B
SCHEMBL18649253 0.61 LMNA (0.48) PDE10ACHRM3PDE4APDE4BPDE4C
Hydrochloric Acid SCHEMBL29974030 0.61 HTR2C (0.34) HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed