SCHEMBL20042731

SCHEMBL20042731

CC1NCc2nc(C3CC3)nc(N3CCC3)c21

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 18/20 0.51
PDE4A P27815 16/20 0.51
PDE4B Q07343 16/20 0.51
PDE4C Q08493 16/20 0.51
PDE4D Q08499 16/20 0.51
PDE10A Q9Y233 2/20 0.44
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM5 P08912 1/20 0.40
CHRM1 P11229 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042736 0.81 NPY5R (0.36) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL20042874 0.81 NPY5R (0.36) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL20042984 0.77 NPY5R (0.35)
SCHEMBL31614998 0.73 MAP2K7 (0.32)
SCHEMBL31614807 0.73 MAP2K7 (0.32)
SCHEMBL20042648 0.72 CHRM3 (0.51) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL20042840 0.70 CHRM3 (0.43) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL4423241 0.68 CHRM3 (1.00) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL20042895 0.66 NPY5R (0.35) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL4421504 0.65 PDE10A (0.94) CHRM3PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed