SCHEMBL20042819

SCHEMBL20042819

Cc1nc(C)c(C)c(N2CCC2)n1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 8/20 0.47
PDE4A P27815 6/20 0.47
PDE4B Q07343 6/20 0.47
PDE4C Q08493 6/20 0.47
PDE4D Q08499 6/20 0.47
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
NPY5R Q15761 4/20 0.41
CYP1A2 P05177 1/20 0.40
PDE10A Q9Y233 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
GBA1 P04062 1/20 0.38
HTR6 P50406 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16117368 0.82 LMNA (0.49) PDE4APDE4BPDE4CPDE4DMAPK1
SCHEMBL13219748 0.76 CHRM3 (0.42) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL26890472 0.74 PDE10A (0.50) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL14685224 0.74 NPY5R (0.46) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL22616920 0.68 OPRM1 (0.42)
SCHEMBL12341499 0.67 HRH4 (0.50) MAPK1L3MBTL1MEN1KMT2ACYP1A2
SCHEMBL27741341 0.67 HSD17B10 (0.44) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL15055333 0.67 CHRM3 (0.46) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL26337498 0.67 GBA1 (0.42) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL77166 0.66 LMNA (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed