SCHEMBL20042858

SCHEMBL20042858

Cc1nc2c(c(N3CCC3)n1)C(C)N(C(=O)C1CCOCC1)C2

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
CNR2 P34972 10/20 0.37
PIK3CD O00329 1/20 0.34
CNR1 P21554 2/20 0.33
GPR55 Q9Y2T6 2/20 0.33
CHRM4 P08173 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
KDM4E B2RXH2 1/20 0.32
IDH1 O75874 1/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
NR4A1 P22736 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042990 0.91 CNR1 (0.37) ALDH1A1PIK3CDCNR1GPR55SMN1; SMN2
Hydrochloric Acid SCHEMBL31614990 0.82 PARP1 (0.34) SMN1; SMN2KDM4ELMNATSHRNR4A1
SCHEMBL20042913 0.81 PREP (0.37) ALDH1A1SMN1; SMN2KDM4ELMNATSHR
SCHEMBL31614760 0.80 SMN1; SMN2 (0.36) SMN1; SMN2KDM4ELMNATSHRNR4A1
SCHEMBL20042840 0.77 CHRM3 (0.43) CHRM4
SCHEMBL20042885 0.77 PIP5K1C (0.38) ALDH1A1SMN1; SMN2KDM4EIDH1LMNA
SCHEMBL20042706 0.77 ALDH1A1 (0.43) ALDH1A1CNR2CNR1GPR55CHRM4
Trifluoroacetic Acid SCHEMBL31615017 0.77 GPR6 (0.32)
SCHEMBL31615046 0.77 HPGD (0.42) ALDH1A1PIK3CDMEN1KMT2A
SCHEMBL31615054 0.77 HPGD (0.42) ALDH1A1PIK3CDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed