SCHEMBL2004334

SCHEMBL2004334

Cc1c(CC(=O)O)c2c(F)c(O)ccc2n1C(=O)c1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 8/20 0.43
AKR1C2 P52895 8/20 0.43
TSHR P16473 2/20 0.43
LMNA P02545 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
NFKB1 P19838 1/20 0.43
HIF1A Q16665 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
PTGS2 P35354 4/20 0.41
PTGS1 P23219 2/20 0.41
ABCB1 P08183 1/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.38
AKR1C4 P17516 1/20 0.38
AKR1C1 Q04828 1/20 0.38
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004418 0.88 PTGS2 (0.46) AKR1C3AKR1C2TSHRLMNACYP1A2
SCHEMBL2007710 0.87 AKR1C3 (0.47) AKR1C3AKR1C2TSHRLMNACYP1A2
SCHEMBL2002963 0.87 LMNA (0.48) AKR1C3AKR1C2TSHRLMNACYP1A2
SCHEMBL5558739 0.83 AKR1C3 (0.57) AKR1C3AKR1C2TSHRLMNACYP1A2
SCHEMBL2002636 0.82 AKR1C3 (0.49) AKR1C3AKR1C2TSHRLMNACYP1A2
SCHEMBL5554171 0.81 AKR1C3 (0.52) AKR1C3AKR1C2TSHRLMNACYP1A2
SCHEMBL3005871 0.81 AKR1C3 (0.64) AKR1C3AKR1C2LMNACYP1A2CYP2D6
SCHEMBL2001676 0.80 LMNA (0.39) AKR1C3AKR1C2TSHRLMNACYP1A2
SCHEMBL5554232 0.80 AKR1C3 (0.52) AKR1C3AKR1C2TSHRLMNACYP1A2
SCHEMBL2004535 0.80 ABCB1 (0.48) AKR1C3AKR1C2TSHRLMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed