SCHEMBL20047071

SCHEMBL20047071

CSc1ccc(-c2ccc3nc(N)ccc3c2)cc1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 15/20 0.65
CTSD P07339 1/20 0.53
NCK1 P16333 1/20 0.51
PLAU P00749 1/20 0.50
NCF1 P14598 4/20 0.47
PIK3CD O00329 1/20 0.42
ABL1 P00519 1/20 0.42
EGFR P00533 1/20 0.42
HCK P08631 1/20 0.42
SRC P12931 1/20 0.42
KDR P35968 1/20 0.42
PIK3CA P42336 1/20 0.42
PIK3CB P42338 1/20 0.42
MTOR P42345 1/20 0.42
PIK3CG P48736 1/20 0.42
EPHB4 P54760 1/20 0.42
PRKDC P78527 1/20 0.42
NOS2 P35228 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22926832 0.79 BACE1 (1.00) BACE1CTSDNCK1PLAUNCF1
SCHEMBL28147640 0.78 ESR1 (0.44)
SCHEMBL10366751 0.78 ADORA1 (0.40) BACE1NCF1PIK3CDPIK3CAPIK3CB
SCHEMBL20047185 0.77 NCF1 (0.75) BACE1CTSDNCK1PLAUNCF1
SCHEMBL7702979 0.74 DYRK1A (0.46)
SCHEMBL5478956 0.71 BACE1 (0.62) BACE1CTSDNCK1PLAUNCF1
SCHEMBL27960721 0.71 BACE1 (0.57) BACE1CTSDNCK1PLAUNCF1
SCHEMBL12260044 0.71 ESR1 (0.42)
SCHEMBL21898203 0.71 ESR1 (0.55)
SCHEMBL20047226 0.70 BACE1 (0.64) BACE1CTSDNCK1PLAUNCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017223514-A9 LXR INVERSE AGONISTS FOR TREATMENT OF CANCER SAINT LOUIS UNIVERSITY (US) 2018-04-12 WO disclosed