SCHEMBL7702979

SCHEMBL7702979

CSc1ccc(-c2cc(N)nc(N)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 16/20 0.46
CDK9 P50750 3/20 0.46
ADORA3 P0DMS8 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
DYRK2 Q92630 1/20 0.42
APP P05067 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31298734 0.79 ADORA3 (0.44) DYRK1ACDK9ADORA3MEN1KMT2A
SCHEMBL27195567 0.77 ADORA3 (0.54) CDK9ADORA3MEN1KMT2AAPP
SCHEMBL2090059 0.77 NOS3 (0.39) DYRK1A
SCHEMBL10528160 0.76 ALDH1A1 (0.50)
SCHEMBL10300271 0.76 ALDH1A1 (0.50)
SCHEMBL7708521 0.76 MEN1 (0.67) DYRK1ACDK9MEN1KMT2ADYRK2
SCHEMBL3790289 0.75 ALDH1A1 (0.58) MEN1KMT2AAPP
SCHEMBL20047071 0.74 BACE1 (0.65)
SCHEMBL13551944 0.74 DYRK1A (0.48) DYRK1ACDK9MEN1KMT2ADYRK2
SCHEMBL28147640 0.73 ESR1 (0.44) ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed