SCHEMBL20048439

SCHEMBL20048439

CCOC(=O)Cc1c(C)[nH]c2cc(B(O)O)ccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.43
LMNA P02545 1/20 0.43
GAA P10253 4/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
KLK6 Q92876 3/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
AKR1C2 P52895 1/20 0.40
HCRTR1 O43613 1/20 0.39
PKM P14618 1/20 0.39
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KLK8 O60259 1/20 0.38
KLK14 Q9P0G3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8291790 0.82 JAK2 (0.47) KDM4ELMNAGAAALDH1A1MAPT
SCHEMBL3394416 0.82 PTGS1 (0.44) KDM4ELMNAGAAALDH1A1MAPT
SCHEMBL1165573 0.78 KDM4E (0.68) KDM4ELMNAGAAALDH1A1MAPT
SCHEMBL31487317 0.78 KDM4E (0.68) KDM4ELMNAGAAALDH1A1MAPT
SCHEMBL8296306 0.76 PRSS1 (0.55) KDM4ELMNAGAAALDH1A1MAPT
SCHEMBL11331437 0.76 KDM4E (0.49) KDM4ELMNAGAAALDH1A1MAPT
SCHEMBL8291738 0.76 KDM4E (0.69) KDM4ELMNAGAAALDH1A1MAPT
SCHEMBL6222629 0.75 GAA (0.63) KDM4ELMNAGAAALDH1A1MAPT
SCHEMBL5190391 0.74 JAK2 (0.55) KDM4ELMNAGAAALDH1A1MAPT
SCHEMBL1191675 0.74 KDM4E (0.51) KDM4ELMNAGAAALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018065607-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2018-04-12 WO disclosed