SCHEMBL2005171

SCHEMBL2005171

CCOc1ccc2c(c1)c(C(=O)c1nnc(-c3cccnc3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.38
MAPK1 P28482 2/20 0.38
HTT P42858 1/20 0.38
F2RL3 Q96RI0 5/20 0.38
RET P07949 1/20 0.36
KDM4E B2RXH2 4/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPT P10636 3/20 0.34
ALOX5AP P20292 2/20 0.34
ALOX5 P09917 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
EDNRB P24530 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004484 0.94 KDM4E (0.38) LMNAF2RL3RETKDM4EALDH1A1
SCHEMBL2002744 0.92 F2RL3 (0.40) LMNAMAPK1F2RL3KDM4EALDH1A1
SCHEMBL2004592 0.92 ALOX5AP (0.41) LMNAMAPK1HTTKDM4EALDH1A1
SCHEMBL2008151 0.92 LMNA (0.39) LMNAMAPK1F2RL3KDM4EALDH1A1
SCHEMBL2010466 0.91 RET (0.38) LMNAMAPK1RETKDM4EALDH1A1
SCHEMBL2006961 0.91 LMNA (0.40) LMNAMAPK1HTTF2RL3KDM4E
SCHEMBL2008130 0.90 ALOX5AP (0.39) LMNAMAPK1HTTF2RL3RET
SCHEMBL2003814 0.90 F2RL3 (0.36) LMNAF2RL3RETKDM4EALDH1A1
SCHEMBL2005825 0.89 RET (0.38) LMNAMAPK1RETKDM4EALDH1A1
SCHEMBL2004562 0.89 RET (0.37) LMNAMAPK1RETKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed