SCHEMBL2004592

SCHEMBL2004592

CCOc1ccc2c(c1)c(C(=O)c1nnc(-c3cccnc3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 7/20 0.41
ALOX5 P09917 3/20 0.41
MAPK1 P28482 2/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
PTGES2 Q9H7Z7 1/20 0.40
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C9 P11712 2/20 0.38
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C19 P33261 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
MAPT P10636 2/20 0.36
NTRK1 P04629 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002122 0.93 PTGES2 (0.41) ALOX5APALOX5MAPK1LMNAPTGES2
SCHEMBL2004616 0.92 ALOX5AP (0.42) ALOX5APALOX5MAPK1LMNACYP3A4
SCHEMBL2005171 0.92 LMNA (0.38) ALOX5APALOX5MAPK1LMNAHTT
SCHEMBL2007666 0.91 MAPK1 (0.43) ALOX5APALOX5MAPK1LMNACYP3A4
SCHEMBL2006720 0.90 ALOX5AP (0.44) ALOX5APALOX5MAPK1LMNAHTT
SCHEMBL2010014 0.90 MAPK1 (0.42) ALOX5APALOX5MAPK1LMNAHTT
SCHEMBL2004532 0.90 PTGES2 (0.42) ALOX5APALOX5MAPK1LMNAHTT
SCHEMBL2002959 0.89 ALOX5AP (0.42) ALOX5APALOX5LMNAPTGES2CYP3A4
SCHEMBL2008741 0.89 PTGES2 (0.44) ALOX5APMAPK1LMNAHTTPTGES2
SCHEMBL2003185 0.88 PTGES2 (0.41) ALOX5APALOX5MAPK1LMNAPTGES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed