SCHEMBL20052448

SCHEMBL20052448

CS(=O)(=O)/C=C/[C@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OCc1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 9/20 0.74
CASP7 P55210 6/20 0.74
CASP1 P29466 5/20 0.74
CASP9 P55211 4/20 0.71
CASP4 P49662 2/20 0.71
CASP5 P51878 2/20 0.71
CASP6 P55212 2/20 0.71
CASP8 Q14790 2/20 0.71
CASP10 Q92851 2/20 0.71
NMBR P28336 2/20 0.56
SIRT5 Q9NXA8 1/20 0.55
MAPT P10636 2/20 0.54
GAA P10253 1/20 0.54
HTT P42858 1/20 0.54
LMNA P02545 1/20 0.53
CA2 P00918 1/20 0.51
MMP9 P14780 1/20 0.51
MMP8 P22894 1/20 0.51
CCKAR P32238 3/20 0.51
CCKBR P32239 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18782323 0.91 CASP3 (0.72) CASP3CASP7CASP1CASP9CASP4
SCHEMBL15462653 0.89 CASP3 (0.92) CASP3CASP7CASP1CASP9CASP4
SCHEMBL19015752 0.86 CASP3 (0.79) CASP3CASP7CASP1CASP9CASP4
SCHEMBL20609292 0.85 CASP3 (1.00) CASP3CASP7CASP1CASP9CASP4
SCHEMBL12829768 0.85 CASP3 (1.00) CASP3CASP7CASP1CASP9CASP4
SCHEMBL18471462 0.85 CASP3 (0.86) CASP3CASP7CASP1CASP9CASP4
SCHEMBL18471954 0.83 CASP3 (0.69) CASP3CASP7CASP1CASP9CASP4
SCHEMBL16376111 0.83 CASP3 (0.92) CASP3CASP7CASP1CASP9CASP4
SCHEMBL20052456 0.82 CASP3 (0.62) CASP3CASP7CASP1CASP9CASP4
SCHEMBL19015930 0.81 CASP3 (0.78) CASP3CASP7CASP1CASP9CASP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9944674-B2 Selective cysteine protease inhibitors and uses thereof GENESIS TECHNOLOGIES LIMITED (BB) 2018-04-17 US disclosed