SCHEMBL20054412

SCHEMBL20054412

O=C(NCc1ncc(-c2ccc(-c3cc4ccc(-c5cnc(CNC(=O)C6CCC(F)(F)CC6)[nH]5)cc4o3)cc2)[nH]1)C1CCC(F)(F)CC1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 9/20 0.49
DYRK1A Q13627 9/20 0.49
WNT1 P04628 7/20 0.39
NR1I2 O75469 1/20 0.38
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
KCNH2 Q12809 3/20 0.36
HTR1A P08908 2/20 0.35
DRD2 P14416 2/20 0.35
DRD4 P21917 2/20 0.35
ROCK2 O75116 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20054476 0.86 GSK3B (0.41) GSK3BDYRK1AWNT1HDAC3HDAC1
SCHEMBL20054480 0.86 GSK3B (0.61) GSK3BDYRK1AWNT1
SCHEMBL20054419 0.85 GSK3B (0.60) GSK3BDYRK1AWNT1HDAC3HDAC1
SCHEMBL15116833 0.81 GSK3B (0.48) GSK3BDYRK1AWNT1NR1I2HDAC3
SCHEMBL20054436 0.80 GSK3B (0.51) GSK3BDYRK1AWNT1HDAC3HDAC1
SCHEMBL20054523 0.79 GSK3B (0.53) GSK3BDYRK1AWNT1HDAC3HDAC1
SCHEMBL20221566 0.79 GSK3B (0.53) GSK3BDYRK1AWNT1HDAC3HDAC1
SCHEMBL20054396 0.79 GSK3B (0.55) GSK3BDYRK1AWNT1HDAC3HDAC1
SCHEMBL20054567 0.79 GSK3B (0.48) GSK3BDYRK1AWNT1HDAC3HDAC1
SCHEMBL20054445 0.79 GSK3B (0.48) GSK3BDYRK1AWNT1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3019196-B1 COMBINATIONS OF HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-06-06 EP disclosed
EP-2802326-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-04-18 EP disclosed