SCHEMBL20054472

SCHEMBL20054472

CC(C)(C)OC(=O)NC(c1ncc(-c2cc3cc4oc(-c5cnc(C(NC(=O)OC(C)(C)C)C(C)(C)C)[nH]5)cc4cc3o2)[nH]1)C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR3 P32745 1/20 0.38
KDM4E B2RXH2 2/20 0.36
GLA P06280 2/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.36
HPGD P15428 2/20 0.36
NR1I2 O75469 1/20 0.34
TRPA1 O75762 2/20 0.34
EPHX2 P34913 2/20 0.33
AAK1 Q2M2I8 3/20 0.32
GABRB1 P18505 1/20 0.32
GABRB2 P47870 1/20 0.32
KMT2A Q03164 1/20 0.32
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
SYK P43405 1/20 0.31
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA9 Q16790 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15116823 1.00 SSTR3 (0.38) SSTR3KDM4EGLAGAAMAPT
SCHEMBL20221549 1.00 SSTR3 (0.38) SSTR3KDM4EGLAGAAMAPT
SCHEMBL16359250 0.88 KMT2A (0.39) SSTR3KDM4EGLAGAAMAPT
SCHEMBL15116835 0.85 NR1I2 (0.43) SSTR3KDM4EGLAGAAMAPT
SCHEMBL20054535 0.82 SSTR3 (0.40) SSTR3KDM4EGLAGAAMAPT
SCHEMBL15116836 0.82 SSTR3 (0.40) SSTR3KDM4EGLAGAAMAPT
SCHEMBL15114363 0.82 NR1I2 (0.42) SSTR3KDM4EGLAGAAMAPT
SCHEMBL20054513 0.78 PRMT5 (0.38) SSTR3KDM4EGLAGAAMAPT
SCHEMBL15116590 0.78 PRMT5 (0.38) SSTR3KDM4EGLAGAAMAPT
SCHEMBL15116624 0.78 SSTR3 (0.44) SSTR3TRPA1EPHX2AAK1SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2802326-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-04-18 EP disclosed