SCHEMBL20055076

SCHEMBL20055076

CCc1ccc2c(c1)N(C)c1ccc(C(C)C)cc1O2

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
NR1H3 Q13133 1/20 0.32
MAPT P10636 1/20 0.31
MIF P14174 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2A6 P11509 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2705592 0.87 NR1H3 (0.36) NR1H3
SCHEMBL13071244 0.81 NR1H3 (0.33) NR1H3
SCHEMBL17656225 0.79 AKR1C3 (0.38) AKR1C3AKR1C2MAPTCYP1A2CYP2A6
SCHEMBL2756740 0.78 NR1H3 (0.33) NR1H3
SCHEMBL1102428 0.76 KDM4E (0.44) NR1H3MAPTMIF
SCHEMBL13892833 0.74 ALDH1A1 (0.41)
SCHEMBL13821481 0.74 NR1H3 (0.34) NR1H3
SCHEMBL13070643 0.72 CYP2D6 (0.43) AKR1C3AKR1C2MAPT
SCHEMBL20055030 0.70 BRD4 (0.33) AKR1C3AKR1C2NR1H3MAPTCYP1A2
SCHEMBL13070864 0.69 TSHR (0.33) AKR1C3AKR1C2MAPTCYP1A2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3309157-A1 ANTIVIRAL COMPOUNDS Gilead Pharmasset LLC (US) 2018-04-18 EP disclosed