SCHEMBL20056161

SCHEMBL20056161

CNCCN1CCC(CNC(=O)c2ccc(C(C)(C)C)cc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.58
LMNA P02545 1/20 0.58
GAA P10253 1/20 0.58
MAPT P10636 1/20 0.58
MAPK1 P28482 1/20 0.58
HTT P42858 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
CACNA1I Q9P0X4 9/20 0.57
KCNH2 Q12809 7/20 0.57
CACNA1H O95180 1/20 0.53
CYP2D6 P10635 1/20 0.53
CARM1 Q86X55 3/20 0.53
PRMT6 Q96LA8 3/20 0.53
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19226529 0.85 NAMPT (0.59) ALDH1A1LMNAGAAMAPTMAPK1
SCHEMBL4280597 0.85 ALDH1A1 (0.52) ALDH1A1LMNAGAAMAPTMAPK1
SCHEMBL19112716 0.84 ALDH1A1 (0.51) ALDH1A1LMNAGAAMAPTMAPK1
SCHEMBL4275124 0.84 ALDH1A1 (0.51) ALDH1A1LMNAGAAMAPTMAPK1
SCHEMBL19113313 0.83 CARM1 (0.56) CACNA1IKCNH2CACNA1HCYP2D6CARM1
SCHEMBL15317662 0.82 MAPK14 (0.57) ALDH1A1LMNAGAAMAPTMAPK1
SCHEMBL19113003 0.81 KCNH2 (0.55) CACNA1IKCNH2CACNA1HCYP2D6CARM1
SCHEMBL17886674 0.80 ALDH1A1 (0.67) ALDH1A1LMNAGAAMAPTMAPK1
SCHEMBL17886696 0.80 ALDH1A1 (0.67) ALDH1A1LMNAGAAMAPTMAPK1
SCHEMBL19112707 0.80 CACNA1I (0.74) CACNA1IKCNH2CACNA1HCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3189839-B1 N-PIPERIDINYL ACETAMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS PRAXIS PREC MEDICINES INC (US) 2020-05-20 EP disclosed
EP-2300007-B1 N-PIPERIDINYL ACETAMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS TARO PHARMACEUTICALS INC (CA) 2018-04-18 EP disclosed