SCHEMBL20056469

SCHEMBL20056469

C=C(N)c1cccc(-c2ccc(O)c(C)c2)c1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 14/20 0.59
HSD17B2 P37059 14/20 0.59
ESR2 Q92731 1/20 0.56
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C19 P33261 2/20 0.46
ERN1 O75460 1/20 0.44
HSD17B14 Q9BPX1 1/20 0.44
APP P05067 1/20 0.41
TLR8 Q9NR97 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19608277 0.83 HSD17B1 (0.59) HSD17B1HSD17B2ESR2CYP3A4CYP2D6
SCHEMBL20056592 0.83 HSD17B1 (0.68) HSD17B1HSD17B2ESR2ERN1HSD17B14
SCHEMBL16581352 0.80 HSD17B1 (0.77) HSD17B1HSD17B2ESR2CYP3A4CYP2D6
SCHEMBL20056514 0.78 HSD17B1 (0.69) HSD17B1HSD17B2ESR2CYP3A4CYP2D6
SCHEMBL28903928 0.78 HSD17B1 (0.69) HSD17B1HSD17B2ESR2ERN1HSD17B14
SCHEMBL29904856 0.78 HSD17B1 (0.69) HSD17B1HSD17B2ESR2ERN1HSD17B14
SCHEMBL20243662 0.76 PRSS1 (0.64)
SCHEMBL272034 0.75 HSD17B1 (0.68) HSD17B1HSD17B2ESR2CYP3A4CYP2D6
SCHEMBL29696046 0.75 HSD17B1 (0.68) HSD17B1HSD17B2ESR2CYP3A4CYP2D6
SCHEMBL29429121 0.75 HSD17B1 (0.68) HSD17B1HSD17B2ESR2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970353-B1 MANNOSE DERIVATIVES FOR TREATING BACTERIAL INFECTIONS VERTEX PHARMA (US) 2018-04-18 EP disclosed