SCHEMBL20060207

SCHEMBL20060207

CN/C(CCc1ccccc1)=C1\C(=N)CC/C(=C\N(C)C)C1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
KDM4E B2RXH2 1/20 0.35
CMA1 P23946 1/20 0.34
ALDH1A1 P00352 4/20 0.32
HDAC2 Q92769 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
GAA P10253 1/20 0.31
ALOX15 P16050 1/20 0.31
KEAP1 Q14145 1/20 0.31
AKR1C3 P42330 1/20 0.30
AKR1C2 P52895 1/20 0.30
ALOX5 P09917 1/20 0.30
EP300 Q09472 1/20 0.30
CARM1 Q86X55 1/20 0.30
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20060208 0.89 KDM4E (0.34) KMT2AMEN1KDM4EALDH1A1SMN1; SMN2
SCHEMBL20059942 0.82
SCHEMBL20060035 0.78 KDM4E (0.36) KMT2AMEN1KDM4EALDH1A1SMN1; SMN2
SCHEMBL20060031 0.76
SCHEMBL20060139 0.75 CMA1 (0.39) CMA1ALDH1A1HDAC2HDAC8HDAC6
SCHEMBL20060212 0.74 MAPT (0.32) KMT2AMEN1KDM4EALDH1A1HPGD
SCHEMBL20060200 0.72 KMT2A (0.45) KMT2AMEN1KDM4EALDH1A1SMN1; SMN2
SCHEMBL20060156 0.71
SCHEMBL20060215 0.70
SCHEMBL20059926 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595987-B1 NEW AMINOPYRAZOLOQUINAZOLINES BOEHRINGER INGELHEIM INT (DE) 2018-04-18 EP disclosed